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Supplements To Help Fall Asleep

Updated: Jun 19

Falling asleep should be as natural and easy as letting gravity pull you down a slide, but sometimes, it isn't. In these cases, the first step in fixing the problem is making sure that you aren't taking something that causes it.



Take a look through your supplements and prescriptions and ask yourself, did the sleep problem start or get worse around the same time that you started a particular supplement or drug? If that's the case, talk with your doctor or prescribing physician about it. Check especially carefully for any folate or methyl donors like methyl folate, methyl B12, SAMe, TMG, and even things that spare methyl groups, like creatine, can be a problem. For some of us, too many methyl groups means you're just not getting to sleep. At all. Ever. So understand your supplements first.


Also, strongly consider anything that has known "upper" potential - ADHD medications, steroids, thyroid medications, and some antidepressants. Even if you've been taking the same dose for years, if your health has changed then your need might also have changed. Often, when people work on their methylation and improve that foundational level of health, then the amount of medication they need decreases.


Next, think about what keeps you awake - is it that your body won't settle down? Your mind? Something mysterious? Let's talk about some options.


Supplements to Relax Your Body


If your body won't relax that almost always means unwanted muscle activity like twitches, zings, pings, crawling feeling, or just discomfort. Of course, do your sleep hygiene. Avoid alcohol before bed, make sure your evening meal is high protein, lower carb, and drink enough water throughout the day. If you have restless legs syndrome, also do some gentle stretching before bed. In terms of supplements, here are my favorites for body relaxation:


  • Magnesium—Magnesium is necessary with restless legs or body tension at night. Magnesium is your natural muscle relaxer, physiologically opposing the calcium that binds to your muscle fibers to help them contract. Magnesium dosing is variable between people and also for each person at different times in their life. The best guide is trial and error; not enough magnesium won't give you the physical relaxation that you're looking for, and too much magnesium will cause a loose stool in the morning. Also, you don't need a fancy form of magnesium. Simple forms like citrate or oxide work just as well for this application as the designer forms. It's rare, but I've seen a few clients over the years who have the opposite reaction to magnesium, and if that is you, try a low-dose calcium chewable at bedtime instead.

  • GABA—GABA is an inhibitory neurotransmitter, meaning that it calms down all of the excess neurological activity to help you calm your body and relax your mind. Standard dosing of GABA for sleep is roughly 300 mg, about an hour before bed. GABA does lower blood pressure for some people, which usually isn't a problem during sleep, but if you have medically low blood pressure, then it's good to talk with your doctor before starting a GABA supplement.

  • Passionflower—This herb has several physically and mentally relaxing properties. It has been shown to gently boost levels of GABA in your brain. It is also mentally calming and soothing and is well known as a supportive herb for sleep and relaxation.


Supplements to Relax Your Mind


An agitated mind is fully capable of overriding all of your good sleep hygiene and keeping you awake at night. Non-supplement techniques like meditation, deep breathing exercises, exercise, and cognitive behavioral therapy are the most effective tools here, but they take time and persistence. While you're building the routine of meditation or CBT, here are some supplements that can help support your progress.


  • Valerian Root—Valerian has well-documented effects on sleep through several mechanisms of action. It raises levels of GABA, which we discussed as a physical and mental relaxant, and also contains unique compounds like valerenic acids and valepotriates, which also contribute to its effectiveness. Valerian helps to improve overall sleep quality and decrease the time it takes to fall asleep. It also reduces feelings of anxiety, as well as some hormone symptoms in women, including PMS and menopausal hot flashes.

  • Bifidobacterium longum 1714—This unique strain of gut bacteria works on the gut-stress connection. In a double-blinded placebo-controlled study, sleep quality and duration improved significantly in participants undergoing exam-related stress after just four weeks of use. This bacterial strain is shown to reduce overall stress response and help normalize morning cortisol levels as well.

  • Aromatherapy—Research has shown that some essential oils can help to promote anxiety relief and better sleep outcomes. Chamomile and lavender are well-documented, and additi.

  • Chamomile—I'm sure at least a few of you had a mother or grandmother prepare chamomile tea for you when you were having a hard time sleeping. Mine certainly did. It turns out that the research shows chamomile to be effective in sleep disorders and generalized anxiety disorder, so your ancestors knew what they were talking about.

  • Glycine—Glycine is a component of protein. It passively diffuses across the blood-brain barrier and modulates neurotransmitters in the braional studies have shown orange and peppermint oil to be beneficin. Three grams before bedtime has been shown to improve sleep quality and decrease the time it takes to get to sleep.


The Miracle of Melatonin - The King of Supplements to Help Fall Asleep


Melatonin is one of my favorite supplements simply because it has so many beneficial functions in the body, and it is your body's natural sleep hormone. Melatonin helps enhance sleep, regulates circadian rhythm, acts as an antioxidant (especially within the brain and spinal cord), boosts immune function, reduces inflammation, slows aging, and has anticancer activities. Outside of that, it's neuroprotective, helps control chronic diseases like cardiovascular disease, diabetes, and obesity. It even helps to regulate mood, sexual maturation, and body temperature.


Natural melatonin is found in plants, animals, and bacteria, and we all get some from food sources daily. Melatonin supplements to help fall asleep are easy to find and generally well tolerated, although some people report more vivid dreams or some sleep-hangover-type feelings in the morning. Doses from 1 - 10 mg are used for sleep, and doses around 20 mg are used as a supportive therapy for solid tumors.


Also, small doses of melatonin can be taken if you wake at night and can't get back to sleep. Some evidence suggests that even if it doesn't bring you back to sleep, it does help your brain to sustain less damage from sleep loss.


Melatonin is a great tool to keep on hand. It can help enhance your sleep quality and get you to sleep faster.


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Please Read: The information here is for educational purposes only. Please consult with your primary care physician before making changes to your diet, supplements, or pharmaceutical medications. If you are having a medical emergency, please call 911. Your life and health are precious.

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